[1] ZHANG Y, ZHANG X L, ZOU Y, et al. Population pharmacokinetics of sirolimus in Chinese adult liver transplant recipients: a retrospective study[J]. Xenobiotica, 2021, 51(12): 1408-1415. doi:  10.1080/00498254.2022.2025628
[2] MATHIYAZHAGAN G, HASAN F, CHAUHAN P, et al. Spondyloenchondrodysplasia with immune dysregulation: Role of sirolimus[J]. Pediatr Blood Cancer, 2022, 69(10): e29672. doi:  10.1002/pbc.29672
[3] MOES D J, GUCHELAAR H J, DE FIJTER J W. Sirolimus and everolimus in kidney transplantation[J]. Drug Discov Today, 2015, 20(10): 1243-1249. doi:  10.1016/j.drudis.2015.05.006
[4] ZHANG X T, CHEN Z Z, TAO C, et al. Effect of surface property on the release and oral absorption of solid sirolimus-containing self-microemulsifying drug delivery system[J]. AAPS PharmSciTech, 2021, 22(3): 108. doi:  10.1208/s12249-021-01978-z
[5] HU X W, LIN C, CHEN D X, et al. Sirolimus solid self-microemulsifying pellets: formulation development, characterization and bioavailability evaluation[J]. Int J Pharm, 2012, 438(1-2): 123-133. doi:  10.1016/j.ijpharm.2012.07.055
[6] JANNIN V, MUSAKHANIAN J, MARCHAUD D. Approaches for the development of solid and semi-solid lipid-based formulations[J]. Adv Drug Deliv Rev, 2008, 60(6): 734-746. doi:  10.1016/j.addr.2007.09.006
[7] O’DRISCOLL C M, GRIFFIN B T. Biopharmaceutical challenges associated with drugs with low aqueous solubility: the potential impact of lipid-based formulations[J]. Adv Drug Deliv Rev, 2008, 60(6): 617-624. doi:  10.1016/j.addr.2007.10.012
[8] 余越, 陶春, 杨海跃, 等. 不同孔径介孔二氧化硅纳米粒的制备及其用于固化西罗莫司自微乳[J]. 药学学报, 2017, 52(6): 985-991.
[9] 黄雯婷, 刘志宏, 张灵娜, 等. 基于介孔硅固化自微乳的西罗莫司缓释片的制备与评价[J]. 药学学报, 2023, 58(4): 1049-1058.
[10] 程晓昆, 仇俊新, 王娅莉, 等. 关于体外溶出实验在仿制药一致性评价中的应用与思考[J]. 中国医药工业杂志, 2019, 5(9): 1065-1071.
[11] 陶春, 陈菊明, 黄爱文, 等. 自微乳缓释片中西罗莫司的稳定性提高研究[J]. 中国医院药学杂志, 2017, 37(17): 1675-1679.
[12]

ZHAO D, FENG J, HUO Q, et al. Triblock copolymer syntheses of mesoporous silica with periodic 50 to 300 angstrom pores[J]. Science, 1998, 279(5350): 548-552. doi:  10.1126/science.279.5350.548
[13] 崔福德. 药剂学[M]. 7版. 北京: 人民卫生出版社, 2011: 420-436.
[14] 潘卫三, 杨星钢. 工业药剂学[M]. 4版. 北京: 中国医药科技出版社, 2019: 533.